TABLE XI

Japanese Pharmaceutical Excipients

NameUsesAdministration Route
Aluminum chloridePotentiating agentIM, SC
Aluminum hydroxideAdsorbentIM, SC
Anhydrous sodium pyrophosphateDispersing agent, Isotonicity, StabilizerIV, IM, intraspinal
Calcium disodium edetateStabilizerIV, SC, intra-arterial, intraspinal, other
Calcium D-saccharateStabilizerIV
CreatinineBuffering agent, StabilizerIV, IM, intracutaneous, SC, other injection
CresolPreservativeIV, IM, SC
L-CystineStabilizerIV
Cysteine hydrochlorideAntioxidant, StabilizerIM, IV
Dibasic sodium citrateBuffering agent, VehicleIV
DiethanolamineBuffer, Solubilizer, StabilizerIV
N, N-DimethylacetamideSolventIV
Disodium hydrogen phosphate, AnhydrousBuffering agent, pH adjustmentIV, SC, IM, other injection
Ethyl oleateSolventIM, intracutaneous
EthylureaSolubilizing agentIM, IV
Ferric chlorideStabilizerIV
GentisylethanolamideAntisepticIV
N-hydroxyethyl lactamide solutionSolubilizing agentIV
InositolStabilizer, VehicleIV, IM
L-Lysine-L-glutamateSolubilizing agent, StabilizerIV
Magnesium gluconateStabilizerIV
Maleic acidBuffering agent, pH adjustment, StabilizerIM
Maleic anhydrideSolubilizer, StabilizerIV
Methanesulfonic acidpH adjustmentIM, SC
DL-MethionineStabilizerIM, intra-arterial, SC, intracutaneous
Monoethanol amineBuffer agent, pH adjustment, Solubilizer, StabilizerIV
Monopotassium L-glutamate monohydratePreservative, StabilizerSC
Oleic acid and purified oleic acidDispersing agent, SolventIV
Oleyl alcoholIV
Phosphoric acidBuffer agent, Isotonicity, pH adjustment, Solubilizing agent, StabilizerIV, IM, SC
Polyoxyethylene castor oil (average added molar ethylene oxide is ∼35)Dispersing agent, Emulsifying agent, Solubilizing agent, Stabilizer, Surfactant, Suspending agent, VehicleIV
Polyoxyethylene hydrogenated castor oil 50Dispersing agent, Emulsifying agent, Solubilizing agentIM, IV
Polyoxyethylene hydrogenated castor oil 60Dispersing agent, Emulsifying agent, Solubilizing agentSC, IM, IV, intraspinal
Polyoxyethylene[160] polyoxypropylene [30] glycolDispersing agent, Emulsifying agent, Solubilizer, Stabilizer, Suspending agent, Vehicle, Surfactant, Wetting agentIV
Polysorbate 20Dispersing agent, Emulsifying agent, Solubilizer, Surfactant, Stabilizer, Suspending agent, Vehicle, Wetting agentIV, SC
Potassium pyrosulfiteStabilizerIV
Sodium acetyl tryptophanStabilizerIV, SC
Sodium caprylateStabilizerIV, SC
Sodium chondroitin sulfateStabilizerIV
Sodium desoxycholateSolubilizing agentIntracutaneous, IV, intraspinal
Sodium dihydrogen phosphate anhydrousBuffer agent, Isotonicity, pH adjustment, StabilizerIV, IM, SC
Sodium dihydrogen phosphate dihydrateBuffer agent, Isotonicity, pH adjustment, StabilizerIM, IV, intra-arterial, SC, intracutaneous, intraspinal, other injection
Sodium formaldehydesulfoxylateStabilizerIV, IM
Sodium metasulfobenzoateStabilizerIV, IM, other injection
Sodium sulfiteAntioxidant, StabilizerIV
Sodium thioglycolateAntioxidant, StabilizerIV, IM, SC
Sodium thiomalateIM
Stannous chlorideReducing agentIV
Succinic acidBuffering agent, pH adjustmentIV
Sulfuric acidBuffering agent, pH adjustmentIM, IV, intra-arterial
alpha-ThioglycerolAntioxidantIV, IM, SC
Thioglycolic acidSolubilizing agent, StabilizerIV, IM, SC
Tribasic sodium phosphateBuffering agent, pH adjustmentIV, IM, SC
TriethanolamineBuffer, pH adjuster, Solubilizing agent, StabilizerIV
Purified yolk lecithinEmulsifierIV
Zinc acetateStabilizerSC
  • IM = intramuscular.

    IV = intravenous.

    SC = subcutaneous.